Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Oxidized ATP (oATP)
A 2',3'-dialdehyde derivative of ATP that is commonly used to affinity label nucleotide sites in enzymes
MilliporeSigma™ Calbiochem™ Methysergide Maleate
An antagonist of the 5-HT2B (pki
MilliporeSigma™ Calbiochem™ GSK-3β Inhibitor XI
The GSK-3β Inhibitor XI, also referenced under CAS 626604-39-5, controls the biological activity of GSK-3β. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ p38 MAP Kinase Inhibitor IV
The p38 MAP Kinase Inhibitor IV, also referenced under CAS 1638-41-1, controls the biological activity of p38 MAP Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ PARP Inhibitor III, DPQ
The PARP Inhibitor III, DPQ, also referenced under CAS 129075-73-6, controls the biological activity of PARP. This small molecule/inhibitor is primarily used for Cell Structure applications.
MilliporeSigma™ Calbiochem™ p38 MAP Kinase Inhibitor VIII
The p38 MAP Kinase Inhibitor VIII, also referenced under CAS 321351-00-2, controls the biological activity of p38 MAP Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ TX-1123
A cell-permeable, reversible, and substrate-competitive arylidene-cyclopentenedione derived tyrphostin that acts as an inhibitor for Src, eEF2-K, and PKA, and EGFR-K/PKC at much higher concentrations.
MilliporeSigma™ Calbiochem™ ATM/ATR Kinase Inhibitor
The ATM/ATR Kinase Inhibitor, also referenced under CAS 905973-89-9, controls the biological activity of ATM/ATR Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Tenovin-1
A cell-permeable benzoylthiourea compound that acts as a reversible inhibitor of class III HDAC sirtuins against SirT2 (IC50 = ≈10 μM).
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MilliporeSigma™ Calbiochem™ Prostaglandin EP2 Receptor Antagonist, TG6-10-1
A cell-permeable, 3-acryl-acrylamide derivative that acts as a highly potent, selective, and competitive antagonist of prostaglandin E2 receptor (EP2, Kb =
MilliporeSigma™ Calbiochem™ PK11195
An isoquinoline carboxamide that acts as a potent ligand for peripheral bezodiazepine receptor (Kd = 20
MilliporeSigma™ Calbiochem™ InSolution™ SU6656
A potent inhibitor of Src-family protein tyrosine kinases
MilliporeSigma™ Calbiochem™ PP2A Activating Ligand, ITH12246
A cell-permeable, relatively non-toxic, 1,8-naphthyridine derived compound that blocks the inhibitory effect of protein phosphatase inhibitors, such as okadaic acid, on protein phosphatase 2A (PP2A)
MilliporeSigma™ Calbiochem™ Transglutaminase 2 Inhibitor, ZDON
A cell-permeable, peptide-based, irreversible inhibitor of transglutaminase 2 (TG2; IC50 = 150nM for recombinant TG2). Reacts with the active site cysteine of TG2.
MilliporeSigma™ Calbiochem™ DNA-PK Inhibitor V
The DNA-PK Inhibitor V, also referenced under CAS 404009-46-7, controls the biological activity of DNA-PK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.